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Reaction Mechanism of Glutamate Carboxypeptidase II Revealed by Mutagenesis, X-ray Crystallography, and Computational Methods | Biochemistry
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RCSB PDB - 3BXM: Structure of an inactive mutant of human glutamate carboxypeptidase II [GCPII(E424A)] in complex with N-acetyl-Asp-Glu (NAAG)
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PDF] Human glutamate carboxypeptidase II inhibition: structures of GCPII in complex with two potent inhibitors, quisqualate and 2-PMPA. | Semantic Scholar
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Reaction Mechanism of Glutamate Carboxypeptidase II Revealed by Mutagenesis, X-ray Crystallography, and Computational Methods | Biochemistry
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IUCr) Human glutamate carboxypeptidase II inhibition: structures of GCPII in complex with two potent inhibitors, quisqualate and 2-PMPA
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Structural characterization of P1'-diversified urea-based inhibitors of glutamate carboxypeptidase II. | Semantic Scholar
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PDF) Structural Insight into the Pharmacophore Pocket of Human Glutamate Carboxypeptidase II | Pavel Majer - Academia.edu
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Structural and biochemical characterization of the folyl‐poly‐γ‐l‐glutamate hydrolyzing activity of human glutamate carboxypeptidase II - Navrátil - 2014 - The FEBS Journal - Wiley Online Library
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Interactions between Human Glutamate Carboxypeptidase II and Urea-Based Inhibitors: Structural Characterization | Journal of Medicinal Chemistry
4LQG: X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a phosphoramidate inhibitor
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RCSB PDB - 4P4E: X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a phosphoramidate inhibitor MP1D
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Structure of glutamate carboxypeptidase II, a drug target in neuronal damage and prostate cancer | The EMBO Journal
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The calcium‐binding site of human glutamate carboxypeptidase II is critical for dimerization, thermal stability, and enzymatic activity - Ptacek - 2018 - Protein Science - Wiley Online Library
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PDF] Human glutamate carboxypeptidase II inhibition: structures of GCPII in complex with two potent inhibitors, quisqualate and 2-PMPA. | Semantic Scholar
![2-MPPA | CAS:254737-29-6 | Selective glutamate carboxypeptidase II (GCP II) inhibitor; orally bioavailable | High Purity | Manufacturer BioCrick 2-MPPA | CAS:254737-29-6 | Selective glutamate carboxypeptidase II (GCP II) inhibitor; orally bioavailable | High Purity | Manufacturer BioCrick](https://www.biocrick.com/media/images/struct/BCC7995.png)
2-MPPA | CAS:254737-29-6 | Selective glutamate carboxypeptidase II (GCP II) inhibitor; orally bioavailable | High Purity | Manufacturer BioCrick
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Glutamate carboxypeptidase II as a model system for designing host–guest units: a theoretical approach - Organic & Biomolecular Chemistry (RSC Publishing) DOI:10.1039/D1OB01209F
2cij - membrane-bound glutamate carboxypeptidase II (GCPII) with bound methionine - Summary - Protein Data Bank Japan
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RCSB PDB - 6FE5: X-ray structure of human glutamate carboxypeptidase II (GCPII) - the E424M inactive mutant, in complex with a inhibitor JHU 2249
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Structural and computational basis for potent inhibition of glutamate carboxypeptidase II by carbamate-based inhibitors - ScienceDirect
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Structure of glutamate carboxypeptidase II, a drug target in neuronal damage and prostate cancer | The EMBO Journal
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